Paper
Synthesis, cytotoxic activity, and fluorescence properties of a set of novel 3-hydroxyquinolin-4(1H)-ones
Published Jun 25, 2014 · Jasna Kadrić, K. Motyka, P. Džubák
Tetrahedron Letters
Q3 SJR score
7
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0
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Abstract
Abstract hidden due to publisher request; this does not indicate any issues with the research. Click the full text link above to read the abstract and view the original source.
In Vitro StudyStudy Snapshot
Novel 3-hydroxyquinolin-4(1H)-one derivatives show promising cytotoxic activity against various cancer cell lines and exhibit fluorescence properties similar to analogous derivatives.
PopulationOlder adults (50-71 years)
Sample size24
MethodsObservational
OutcomesBody Mass Index projections
ResultsSocial networks mitigate obesity in older groups.
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References
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Citations
Phosphine-Mediated Redox Cyclization of 1-(2-Nitroaryl)prop-2-ynones to 3-Hydroxyquinolin-4-ones: Formal Intramolecular Oxyamination of α,β-Ynones.
Phosphine-mediated redox transformation of 1-(2-nitroaryl)prop-2-ynones to 3-Hydroxyquinolin-4-ones enables the synthesis of 3-HQs under neutral conditions, making it useful for the total synthesis of japonine and rare quinoline derivative
2022·3citations·Lona Dutta et al.·Organic letters
Organic letters
Fluorinated derivatives of 2-phenyl-3-hydroxy-4(1H)-quinolinone as tubulin polymerization inhibitors.
Fluorinated 2-phenyl-3-hydroxy-4(1H)-quinolinone derivatives show anticancer activity and inhibit microtubule formation, suggesting potential as cancer cell inhibitors.
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European journal of medicinal chemistry
Use of Phenacyl Thiosalicylates for the Preparation of 3-Hydroxybenzo[b]thiophene Derivatives
Phenacyl thiosalicylates can be used to synthesize 3-hydroxybenzo[b]thiophene derivatives, with potential applications in pharmaceutical and nutraceutical industries.
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Synthesis of 2-alkenyl-3-hydroxyquinolin-4(1H)-ones as promising antimicrobial and fluorescent agents
2-Alkenyl-3-hydroxyquinolin-4(1H)-ones show promising antimicrobial and fluorescent properties against specific bacteria, with high excitation wavelengths and well-separated emission bands.
2018·8citations·R. Horak et al.·Tetrahedron
Tetrahedron
Inhibition of Na+/K+-ATPase by 5,6,7,8-tetrafluoro-3-hydroxy-2-phenylquinolin-4(1H)-one.
TFHPQ is an efficient inhibitor of Na+/K+-ATPase, particularly effective at higher concentrations of K+, with a binding site near the cytoplasmic C-terminus.
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