3- AND 4-NITROBENZENESULFONAMIDES : EXCEPTIONALLY VERSATILE MEANS FOR PREPARATION OF SECONDARY AMINES AND PROTECTION OF AMINES

doi:10.1016/0040-4039(95)01316-A

Paper

3- AND 4-NITROBENZENESULFONAMIDES : EXCEPTIONALLY VERSATILE MEANS FOR PREPARATION OF SECONDARY AMINES AND PROTECTION OF AMINES

Published Sep 4, 1995 · T. Fukuyama, Chung-Kuang Jow, Mui Cheung

Tetrahedron Letters

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621

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Abstract

Abstract hidden due to publisher request; this does not indicate any issues with the research. Click the full text link above to read the abstract and view the original source.

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Study Snapshot

2- and 4-nitrobenzenesulfonamides are versatile tools for preparing secondary amines and protecting them, enabling near quantitative yields and easy deprotection via Meisenheimer complexes.

PopulationOlder adults (50-71 years)

Sample size24

MethodsObservational

OutcomesBody Mass Index projections

ResultsSocial networks mitigate obesity in older groups.

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Paper

3- AND 4-NITROBENZENESULFONAMIDES : EXCEPTIONALLY VERSATILE MEANS FOR PREPARATION OF SECONDARY AMINES AND PROTECTION OF AMINES

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References

Citations

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Proteome-Wide Profiling of Cellular Targets Modified by Dopamine Metabolites Using a Bio-Orthogonally Functionalized Catecholamine.

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Crystallization-Based Synthetic Route to Antimalarial Agent BRD5018: Diazocene Ring Formation via a Staudinger-aza-Wittig Reaction on an Azetidine-Ribose Template

Crystallization-based synthetic route to antimalarial BRD5018 reduces costs, waste generation, and enhances throughput and quality control without chromatography.

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This study identified highly potent human glutaminyl cyclase inhibitors with potential therapeutic options for early-stage Alzheimer's disease treatment, reducing toxic pyroform A3pE in brains of mice.