Synthesis and ABCG2 inhibitory evaluation of 5-N-acetylardeemin derivatives.

doi:10.1016/j.bmc.2015.03.017

Paper

Synthesis and ABCG2 inhibitory evaluation of 5-N-acetylardeemin derivatives.

Published May 1, 2015 · Daigo Hayashi, Naoki Tsukioka, Yutaka Inoue

Bioorganic & medicinal chemistry

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Abstract

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In Vitro Study

Study Snapshot

5-N-acetylardeemin derivatives show stronger inhibitory effects on breast cancer resistance protein ABCG2, with the most potent activity observed in the derivative 1m with a 4-tolyl substituent at C-13.

PopulationOlder adults (50-71 years)

Sample size24

MethodsObservational

OutcomesBody Mass Index projections

ResultsSocial networks mitigate obesity in older groups.

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Synthesis and ABCG2 inhibitory evaluation of 5-N-acetylardeemin derivatives.

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