G. Whitlock, J. Blagg, P. Fish
Jan 15, 2008
Citations
0
Influential Citations
21
Citations
Journal
Bioorganic & medicinal chemistry letters
Abstract
A novel series of 1-(2-phenoxyphenyl)methanamines is disclosed, which possess selective dual 5-HT and NA reuptake pharmacology. Analogues with good human in vitro metabolic stability, hERG selectivity and passive membrane permeability were identified.