J. Spencer, A. Burd, C. Goodwin
Feb 18, 2002
Citations
0
Influential Citations
18
Citations
Journal
Tetrahedron
Abstract
Abstract The synthesis of 2-mercapto- and 2-piperazino- (methyl-phenyl)-4,4,5,5-tetramethyl-[1,3,2]dioxaborolanes 4 and 5 , respectively, is described and their inhibitory activity against serine proteases including thrombin was measured. Some of these compounds were studied in both the solid state and in solution, displaying no S–B coordination and only weak N–B coordination.