V. Cecchetti, F. Schiaffella, O. Tabarrini
Mar 6, 2000
Citations
1
Influential Citations
35
Citations
Quality indicators
Journal
Bioorganic & medicinal chemistry letters
Abstract
A series of compounds having a piperazine moiety variously linked to the benzothiazine nucleus were synthesized and evaluated for their in vitro alpha-adrenoceptor affinity by radioligand receptor binding assays. Some compounds bearing a oxyalkyl-(2-methoxyphenyl)piperazine side chain were good alpha1-adrenoreceptor ligands.