Aleksandr V. Denisenko, Andrey P. Mityuk, O. Grygorenko
Aug 26, 2010
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0
Influential Citations
13
Citations
Journal
Organic letters
Abstract
An efficient two-step multigram synthesis of the previously unknown 3-benzyl-3-azabicyclo[3.1.1]heptan-6-one is described. The compound is shown to be a promising building block for further selective derivatization of the cyclobutane ring providing novel conformationally restricted piperidine derivatives.