S. V. Goswami, P. B. Thorat, Mahesh V. Shukla
Apr 1, 2015
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Journal
Research on Chemical Intermediates
Abstract
Abstract3-Chlorophenylboronic acid promotes efficient synthesis of 3-substituted indole derivatives via aza-Friedel–Crafts reaction of indoles, aromatic aldehydes, and N,N-dimethylaniline at room temperature. The mild reaction conditions, excellent yields, and easy experimental workup are striking features of this procedure for synthesis of 3-substituted indoles.