Saurav Bera, P. S. Kandiyal, R. Ampapathi
Mar 11, 2014
Citations
0
Influential Citations
1
Citations
Journal
Synlett
Abstract
Abstract Trifluoroacetic acid catalyzed condensation of aromatic amines with substituted benzaldehydes followed by intramolecular cyclization furnishes a highly effective synthesis of amino acid derived 2,3-dihydro-1H-1,5-benzodiazepines. The strategy provides an efficient access to a library of benzodiazepines that can be explored for potential pharmaceutical or biological activities.