D. Albanese, D. Landini, M. Penso
Apr 22, 2010
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0
Influential Citations
13
Citations
Journal
Organic Process Research & Development
Abstract
A novel, straightforward synthesis of enantiomerically pure 2,6-disubstituted morpholines has been developed. The ring-opening of epoxides with TsNHBoc under solid−liquid phase transfer catalysis conditions occurred with N → O migration of the Boc group, affording an intermediate carbonate that has been easily transformed to morpholines.