N. Mishra, Mijin Jeon, Yongguk Oh
Feb 1, 2017
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Influential Citations
34
Citations
Journal
Organic chemistry frontiers
Abstract
The pyrimidinyl-directed C–H functionalization of indolines with anthranils as amination sources under rhodium(III) catalysis is described. This transformation efficiently provides a range of C7-aminated indoline derivatives with excellent site-selectivity and functional group compatibility. The resulting framework containing amino and carbonyl groups provides facile access to an important synthetic building block, which can be readily converted to biologically interesting heterocycles.