I. Creese, D. Burt, SolomonH Snyder
Apr 30, 1976
Citations
21
Influential Citations
1,989
Citations
Quality indicators
Journal
Science
Abstract
Tritiated haloperidol and tritiated dopamine label postsynaptic dopamine receptors in mammalian brain. Clinical potencies of butyrophenones, phenothiazines, and related drugs correlate closely with their ability to inhibit tritiated haloperidol binding. These binding methods provide a simple in vitro means for evaluating new drugs as potential antischizophrenic agents.