J. Bermudez, F. King, G. Sanger
Dec 1, 1992
Citations
0
Influential Citations
5
Citations
Quality indicators
Journal
Bioorganic & Medicinal Chemistry Letters
Abstract
Abstract The synthesis and 5-HT3 receptor antagonist activity of imidazole derivatives of 3-keto-indazoles, and 3,3-dimethylindolin-1-yl and o-methoxyphenyl amides is described. Results demonstrate that indazole and indoline are effective bioisosteres in the imidazole class of 5-HT3 receptor antagonists.