K. Goerlitzer, S. Herbig, R. D. Walter
Dec 16, 1997
Citations
0
Influential Citations
23
Citations
Journal
ChemInform
Abstract
The 2-acyl-3-aminoindenes 1 and 2 react with formamidine acetate to yield the indeno[1,2-d]pyrimidines 3 and 4. The 4-chloropyrimidine 5, synthesized from 4 with phosphorous oxychloride, reacts with N-nucleophiles to form the title compounds 6-8. Only 8 shows a weak antimalaria activity