D. Boschelli, D. Powell, Jennifer M. Golas
Sep 15, 2003
Citations
0
Influential Citations
10
Citations
Journal
Bioorganic & medicinal chemistry letters
Abstract
4-(2,4-Dichloro-5-methoxy)anilino-5,10-dihydropyrimido[4,5-b]quinolines are potent inhibitors of Src kinase and Src cellular activity while having no effect on Fyn cellular activity. The corresponding 4-(2,4-dichloro-5-methoxy)anilino-pyrimido[4,5-b]quinolines are much less effective Src inhibitors.