Augustin Peneau, Quentin Tricart, C. Guillou
Jun 5, 2018
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0
Influential Citations
6
Citations
Journal
Chemical communications
Abstract
Azepinone derivatives are important frameworks of several natural products and bioactive compounds. They are synthetized using a Rh(iii)-catalyzed intramolecular annulation of benzamide-tethered allylic alcohols. The reaction requires mild conditions at room temperature and affords diversely substituted azepinones bearing a quaternary carbon.