V. Valenta, M. Vlková, J. Holubek
1990
Citations
0
Influential Citations
2
Citations
Journal
Collection of Czechoslovak Chemical Communications
Abstract
Heating ethyl 5-sulfamoyl-2-methoxybenzoate with a series of twelve 3-(tert.amino)propylamines (IIIa-IIIl) afforded the title compounds IIa-IIl which were transformed to salts and subjected to pharmacological screening as potential neuroleptics of the sulpiride series. Only compounds IId (hydrogen oxalate, VUFB-15453) and IIg (methanesulfonate, VUFB-15397) showed indications of the desired psychotropic activity