M. Surman, M. Mulvihill, Marvin J Miller
Jan 10, 2002
Citations
0
Influential Citations
37
Citations
Journal
Organic letters
Abstract
[reaction: see text] N(4)-Hydroxy-1,4-benzodiazepines were synthesized in a single step from synthetically versatile acylnitroso-derived hetero-Diels-Alder cycloadducts. The efficiency of this transformation was found to be dependent on the NH pK(a) of the cycloadduct sulfonamide.