H. Stefani, Stanley N. S. Vasconcelos, Frederico B. Souza
Oct 23, 2013
Citations
0
Influential Citations
15
Citations
Journal
Tetrahedron Letters
Abstract
A general and efficient reaction of indole with oxalyl chloride and nucleophiles providing indole-3-glyoxyl derivatives has been developed in mild conditions. In the same fashion, the other reaction involved the addition of organic azides leading to the synthesis of indole-3-glyoxyl-1,2,3-triazoles, which proceeds smoothly generating the products in moderate to high yields.