A. Armstrong, L. Jones, Jamie D. Knight
Jan 20, 2005
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Influential Citations
70
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Quality indicators
Journal
Organic letters
Abstract
Electrophilic amination of primary aliphatic and aromatic amines is reported using a diethylketomalonate-derived oxaziridine to afford the corresponding N-Boc hydrazines in good to excellent yields. The method allows a one-pot synthesis of pyrazoles from primary amines. [Reaction: see text]