Q. Ding, C. Ye, S. Pu
Jan 14, 2014
Citations
0
Influential Citations
41
Citations
Journal
Tetrahedron
Abstract
An efficient protocol was developed for regio-selective Pd-catalyzed direct ortho-fluorination of 2-arylbenzo[d]thiazoles using N-fluorobenzenesulfonimide (NFSI) as the F+ source, and l-proline as the crucial promoter. The present method offered a practical route to synthesize valuable fluorinated products, which are of potential importance in the pharmaceutical and agrochemical industries.