D. Petrillo, Dale R. Mowrey, S. Allwein
Feb 22, 2012
Citations
0
Influential Citations
9
Citations
Journal
Organic letters
Abstract
Fmoc-O-benzyl-l-phosphoserine is an important building block in the synthesis of Forigerimod, a phosphopeptide being investigated for Systemic Lupus Erythematosus (SLE). An efficient one-pot process was developed using inexpensive, readily available starting materials. This general procedure was used to prepare a variety of protected phosphoamino acids.