Woongki Kim, J. Dannaldson, K. Gates
Jul 22, 1996
Citations
3
Influential Citations
29
Citations
Journal
Tetrahedron Letters
Abstract
Abstract Reaction of 3 H -1,2-benzodithiol-3-one 1-oxide with primary amines or anilines provides reasonable yields (40–70%) of the corresponding 1,2-benzisothiazolin-3(2 H )-ones. These reactions may have relevance to the biological chemistry of 1,2-dithiolan-3-one 1-oxides and also offer a new method for the preparation of certain 1,2-benzisothiazolin-3(2 H )-ones.