L. Malins, Andrew M. Giltrap, Luke J. Dowman
Apr 10, 2015
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0
Influential Citations
31
Citations
Journal
Organic letters
Abstract
The efficient synthesis of a β-thiol phenylalanine derivative is described starting from Garner's aldehyde. The utility of this amino acid in peptide ligation-desulfurization chemistry is described, including the trifluoroethanethiol (TFET)-promoted one-pot assembly of the 62 residue peptide hormone augurin.