S. Schneller, Jiann-Kuan Luo, R. Hosmane
Jul 1, 1984
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Influential Citations
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Journal
Journal of Heterocyclic Chemistry
Abstract
The synthesis of 1-methyl- (1a) and 1-benzyl-6-amino-1H-pyrrolo[3,2-c]pyridin-4(5H)-one (1b) from the appropriate N-alkylaminoacetaldehyde is described. These provide examples of a synthetic procedure that can be used to prepare 1-substituted 6-amino-1H-pyrrolo[3,2-c]pyridin-4(5H)-ones wherein the N-1 substituent is regiospecifically placed.