Jie Wang, Lili Wang, Shanyan Guo
Jun 22, 2017
Citations
1
Influential Citations
30
Citations
Journal
Organic letters
Abstract
An efficient Rh(III)-catalyzed C-H activation protocol has been developed for the synthesis of 2,3-benzodiazepines with use of N-Boc hydrazones and diazoketoesters as substrates. The reaction features retention of the C═N and N-N bonds and selective cleavage of the N-Boc moiety.