Guo-Bo Deng, Zhiqiang Wang, Ren‐Jie Song
Jul 5, 2011
Citations
0
Influential Citations
6
Citations
Journal
Chemical communications
Abstract
A new palladium-catalyzed C-H bond activation-annulation-amination tandem method was presented for selectively synthesizing 3-(aminomethylene)-2-oxoindolines. In the presence of Pd(dba)(2), xantphos (L8), AgOAc and Na(2)CO(3), a variety of 3-chloro-2-iodo-N-arylacrylamides underwent the reaction with amides or amines to afford the corresponding 3-(aminomethylene)-2-oxoindolines in moderate to good yields.