R. Deprez-Poulain, Julie Charton, Virginie Leroux
Nov 12, 2007
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0
Influential Citations
18
Citations
Journal
Tetrahedron Letters
Abstract
We report here the convenient synthesis of 4H-1,2,4-triazole-3-thiols using di-2-pyridyl-thionocarbonate as the thiocarbonyl transfer reagent. This method is suitable for microplate parallel synthesis and produces samples in screening-ready condition. It uses two large sets of building-blocks: amines and hydrazides.