K. Yeung, N. Meanwell
Jul 23, 1998
Citations
0
Influential Citations
10
Citations
Journal
Tetrahedron Letters
Abstract
Abstract 4-Thiomethylbenzisothiazolone-1,1-dioxides were synthesized via the corresponding 4-methylbenzisothiazolone-1,1-dioxides by a regioselective benzylic bromination, followed by conversion of the bromide to the thiol moiety under mild and neutral reaction conditions using 1-(2-hydroxyethyl)-4,6-diphenylpyridine-2-thione (HDPT).