Kazunao Ishiyama, Y. Yamada
Feb 7, 2005
Citations
0
Influential Citations
5
Citations
Journal
Tetrahedron Letters
Abstract
Abstract 7-Hydroxyindole, the key building block for the synthesis of AJ-9677 1 , was prepared from indoline in six steps in 36% overall yield. AJ-9677 1 is a potent and selective adrenaline β3-agonist being considered as a clinical candidate to treat obesity in those who are suffering from diabetes.