Mina Saeedi, M. Mahdavi, A. Foroumadi
Apr 22, 2013
Citations
0
Influential Citations
54
Citations
Journal
Tetrahedron
Abstract
Abstract Using 2-azidobenzaldehyde and propargylamine in a Ugi–Smiles coupling gave easy access to 4,5-dihydro-1,2,3-triazolo[1,5- a ][1,4]benzodiazepine derivatives. This novel approach is based on the reaction between 2-azidobenzaldehyde, propargylamine, isocyanides, and nitrophenols in methanol under reflux conditions without using additional reagents or catalysts.