Ferdinand S. Melkonyan, A. Karchava, M. Yurovskaya
May 10, 2008
Citations
0
Influential Citations
45
Citations
Journal
The Journal of organic chemistry
Abstract
A variety of N-alkylated and N-arylated derivatives of methyl 1 H-indole-3-carboxylate were synthesized efficiently via Ullmann-type intramolecular arylamination, using the CuI-K 3PO 4-DMF system. This catalytic amination procedure can be performed with good to high yields under mild conditions under an air atmosphere.