D. S. Torok, H. Ziffer
Feb 6, 1995
Citations
0
Influential Citations
28
Citations
Journal
Tetrahedron Letters
Abstract
Abstract 11-Azaartemisinin was prepared in 45% yield in a one pot, two-step sequence from the reaction of artemisinin with excess ammonia followed by acid treatment. Analogous reactions of artemisinin with primary alkylamines gave N-alkylazaartemisinins in similar yields.